It binds within the internal cavity of HIF-2α PAS-B (Kd of 81 nM) and disrupts heterodimerization of the full-length HIF-2 transcription factor
Smiles: CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1C=CC(=CC=1)C1SC=NC=1C)C(C)(C)C
Specifically
The synthetic agonist peptides mimicking the tethered ligand of PAR2
791:560-568
Genipin 1-β-D-gentiobioside Size:Contact [email protected] for quotation It binds within the internalGenipin 1 D gentiobioside (Genipin 1 gentiobioside) is one of the most abundant and bioactive iridoid glycosides in Gardenia jasminoides Ellis, which possesses hepatoprotective, anti inflammatory, antioxidant, and antithrombotic activities. Product information CAS Number: 29307 60 6 Molecular Weight: 550. 51 Formula: C23H34O15 Chemical Name: methyl (1S,4aS,7aS) 4a,7a dihydrogenio 1 {[(2S,3R,4S,5S,6R) 2 hydrogenio 3,4,5 trihydroxy 6 ({[(2R,3R,4S,5S,6R)